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BGC
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IUPAC-Bezeichnung
CAS
EINECS
Formel
Inhibitor
Ovoinhibitor
62449-23-4
CDK inhibitor
468740-43-4
C
2
5
H
2
6
ClN
5
O
3
Syk Inhibitor
622387-85-3
C
1
8
H
1
5
N
3
O
3
S
JNK inhibitor
1408064-71-0
C
2
8
H
2
7
N
7
O
2
ERK Inhibitor
1049738-54-6
C
1
4
H
1
6
N
2
O
3
S HCl
Erk inhibitor
294675-79-9
C
1
4
H
1
6
N
2
O
3
S.HCl
UV inhibitors
Wax inhibitor
Inhibitor 702
Inhibitor 701
PKR Inhibitor
608512-97-6
C
1
3
H
8
N
4
OS
uPA Inhibitor
149732-36-5
C
9
H
7
IN
2
Sâ¢HCl
Hcv inhibitor
442666-98-0
C
1
7
H
1
1
ClF
2
N
4
O
2
S
Lck Inhibitor
213743-31-8
C
2
3
H
2
2
N
4
O
PKG Inhibitor
82801-73-8
C
3
8
H
7
4
N
1
8
O
1
0
JAK inhibitor
1187594-09-7
C
1
6
H
1
7
N
7
O
2
S
Akt inhibitor
1004990-28-6
C
2
0
H
2
2
F
2
N
6
O
Itk inhibitor
439574-61-5
C
3
1
H
3
9
N
5
O
4
S
2
Lck inhibitor
847950-09-8
C
3
1
H
3
0
N
8
O
Mek inhibitor
334951-92-7
C
2
6
H
2
6
N
4
O
2
Ros inhibitor
330997-95-0
Cdk4 Inhibitor
546102-60-7
C
2
0
H
1
0
BrN
3
O
2
MDM2 Inhibitor
562823-84-1
C
1
5
H
1
2
BIO
3
IP3K Inhibitor
519178-28-0
C
2
0
H
1
6
F
3
N
7
O
2
EGFR Inhibitor
879127-07-8
C
2
1
H
1
8
F
3
N
5
O
Rock inhibitor
129830-38-2
C
1
4
H
2
1
N
3
O.2HCl
Wee1 Inhibitor
622855-37-2
C
2
0
H
1
1
ClN
2
O
3
Ikkb inhibitor
406209-26-5
C
2
1
H
2
4
N
4
O
2
.HCl
NFAT Inhibitor
249537-73-3
C
7
5
H
1
1
8
N
2
0
O
2
2
S
Chk2 Inhibitor
724708-21-8
C
1
5
H
1
3
N
5
O
2
HDAC inhibitor
660847-06-3
C
2
8
H
3
9
N
5
O
7
Cdk1 Inhibitor
220749-41-7
C
1
7
H
1
1
ClN
2
O
HDAC inhibitor
1026295-98-6
C
2
8
H
3
6
F
3
N
5
O
7
PKCb Inhibitor
257879-35-9
C
2
4
H
2
1
N
5
O
2
Coke inhibitor
IL-8 Inhibitor
138559-60-1
C
4
5
H
6
6
N
1
8
O
7
S
Rock inhibitor
331752-47-7
C
1
4
H
2
1
N
3
O.2HCl.H
2
O
MK2a Inhibitor
41179-33-3
C
2
2
H
2
0
FNO
2
MNK1 Inhibitor
522629-08-9
C
1
1
H
9
FN
6
PknG Inhibitor
329221-38-7
C
1
3
H
1
6
N
2
O
2
S
PDK1 inhibitor
1001409-50-2
C
2
8
H
2
2
F
2
N
4
O
4
FGFR inhibitor
848318-25-2
C
1
8
H
1
5
N
2
O
4
.Na
Cdk9 inhibitor
1415559-43-1
C
2
6
H
2
1
N
5
O
4
S
PGD2-inhibitor
885066-67-1
CETP inhibitor
1149362-88-8
C
3
4
H
4
0
F
6
N
6
O
4
Tak1 inhibitor
1326712-16-6
PKM2 Inhibitor
94164-88-2
Ahas inhibitor
219793-45-0
C
1
9
H
1
2
ClNO
6
S
Cd4k Inhibitor
546102-60-7
C
2
0
H
1
0
BrN
3
O
2
ROCK inhibitor
867017-68-3
C
1
8
H
1
3
ClF
2
N
6
O
IRAK inhibitor
1042224-63-4
C
1
7
H
1
9
N
5
Pi3k inhibitor
1202884-94-3
C
3
1
H
3
5
F
3
N
8
O
3
Mtor inhibitor
1207358-59-5
C
2
5
H
3
0
N
8
O
2
Isoinhibitor k
56094-10-1
Pik-inhibitors
371934-59-7
C
1
9
H
1
7
N
5
O
2
Trka inhibitor
388626-12-8
Pdhk inhibitor
243982-58-3
Srpk inhibitor
218156-96-8
C
1
8
H
1
8
F
3
N
3
O
Jak3 inhibitor
211555-04-3
C
1
6
H
1
4
BrN
3
O
3
ACC2 Inhibitor
SCD1 Inhibitor
Kdm5-inhibitor
Chk1 inhibitor
2097938-64-0
JNK Inhibitor V
345987-15-7
C
2
0
H
1
6
N
6
S
HDAC6 Inhibitor
1045792-66-2
C
2
2
H
3
0
N
4
O
6
PTP1B Inhibitor
765317-72-4
C
2
6
H
1
9
Br
2
N
3
O
7
S
3
c-FMS inhibitor
885704-21-2
C
2
3
H
3
0
N
6
O
Bcl-2 Inhibitor
383860-03-5
C
1
6
H
1
6
N
2
O
4
MMP-3InhibitorI
158841-76-0
C
2
7
H
4
6
N
1
0
O
9
S
Akt Inhibitor X
925681-41-0
C
2
0
H
2
5
ClN
2
O.HCl
Rac1 inhibitory
PTP Inhibitor I
2491-38-5
219-655-0
C
8
H
7
BrO
2
Fabp4 inhibitor
300657-03-8
C
3
1
H
2
6
N
2
O
3
MMP inhibitor 1
124168-73-6
C
2
3
H
3
4
N
6
O
6
PRL-3 Inhibitor
893449-38-2
C
1
7
H
1
1
Br
2
NO
2
S
2
JAK Inhibitor I
457081-03-7
C
1
8
H
1
6
FN
3
O
sPLA2 inhibitor
393569-31-8
C
3
1
H
3
7
NO
4
CaMKP Inhibitor
52789-62-5
258-185-0
C
1
0
H
8
NNaO
7
S
2
Acid inhibitors
MMP Inhibitor V
223472-31-9
C
2
2
H
2
8
N
2
O
6
Flt-3 Inhibitor
301305-73-7
C
1
8
H
2
0
N
2
O
4
S
Stat5 inhibitor
285986-31-4
C
1
6
H
1
1
N
3
O
3
HIF-1 Inhibitor
934593-90-5
C
2
6
H
2
9
NO
5
B-Raf inhibitor
1021950-26-4
C
3
1
H
3
1
FN
6
O
5
B-Raf inhibitor
918505-61-0
C
2
2
H
1
8
F
2
N
4
O
3
S
Scale inhibitor
Ido inhibitor 1
1204669-37-3
C
1
1
H
1
3
BrFN
7
O
4
S
Src Inhibitor 1
179248-59-0
C
2
2
H
1
9
N
3
O
3
ACSS2 inhibitor
ALK inhibitor 1
761436-81-1
C
2
3
H
2
8
BrN
7
O
3
S
B-Raf inhibitor
1315330-11-0
C
2
9
H
3
1
F
3
N
6
O
2
ALK inhibitor 2
761438-38-4
C
2
3
H
2
8
ClN
7
O
3
S
Scd inhibitor 1
1150701-66-8
Plpro inhibitor
1093070-14-4
C
2
2
H
2
2
N
2
O
2
MAT2A inhibitor
2201057-10-3
Lck inhibitor 2
944795-06-6
C
1
8
H
1
7
N
5
O
2
Btk inhibitor 1
1412418-47-3
K-ras inhibitor
1469338-01-9
C
2
0
H
3
0
ClN
3
O
2
S
3
Akt inhibitor 2
1313881-70-7
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