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IUPAC名
CAS
EINECS
公式
Imatinib
152459-95-5
C
2
9
H
3
1
N
7
O
Apatinib
1218779-75-9
C
2
4
H
2
3
N
5
O.CH
4
O
3
S
Icotinib
610798-31-7
C
2
2
H
2
1
N
3
O
4
Apatinib
1275609-10-3
Axitinib
319460-85-0
C
2
2
H
1
8
N
4
OS
Afatinib
439081-18-2
C
2
4
H
2
5
ClFN
5
O
3
Afatinib
850140-72-6
C
2
4
H
2
5
ClFN
5
O
3
Apatinib
811803-05-1
C
2
4
H
2
3
N
5
O
Avitinib
1557267-42-1
Icotinib
1204313-51-8
C
2
2
H
2
1
N
3
O
4
.HCl
Dovitinib
915769-50-5
C
2
1
H
2
1
FN
6
O.C
3
H
6
O
3
.H
2
O
Dovitinib
405169-16-6
C
2
1
H
2
1
FN
6
O
Dovitinib
804551-71-1
Ponatinib
943319-70-8
C
2
9
H
2
7
F
3
N
6
O
Sapitinib
848942-61-0
C
2
3
H
2
5
ClFN
5
O
3
Ibrutinib
936563-96-1
C
2
5
H
2
4
N
6
O
2
Tepotinib
1100598-32-0
C
2
9
H
2
8
N
6
O
2
Bafetinib
887650-05-7
C
3
0
H
3
1
F
3
N
8
O
Volitinib
1313725-88-0
C
1
7
H
1
5
N
9
Erlotinib
183321-74-6
C
2
2
H
2
3
N
3
O
4
Lapatinib
231277-92-2
C
2
9
H
2
6
ClFN
4
O
4
S
Orantinib
252916-29-3
C
1
8
H
1
8
N
2
O
3
Foretinib
849217-64-7
C
3
4
H
3
4
F
2
N
4
O
6
Masitinib
790299-79-5
C
2
8
H
3
0
N
6
OS
Bafetinib
859212-16-1
C
3
0
H
3
1
N
8
OF
3
Gefitinib
184475-35-2
C
2
2
H
2
4
ClFN
4
O
3
Famitinib
945380-27-8
Sunitinib
557795-19-4
C
2
2
H
2
7
FN
4
O
2
Telatinib
75747-14-7
C
3
1
H
4
3
N
3
O
8
Pelitinib
257933-82-7
C
2
4
H
2
3
ClFN
5
O
2
Dasatinib
302962-49-8
C
2
2
H
2
6
ClN
7
O
2
S
Bosutinib
380843-75-4
C
2
6
H
2
9
Cl
2
N
5
O
3
Neratinib
698387-09-6
C
3
0
H
2
9
ClN
6
O
3
Alectinib
1256580-46-7
C
3
0
H
3
4
N
4
O
2
Henatinib
1239269-51-2
Nilotinib
641571-10-0
C
2
8
H
2
2
F
3
N
7
O
Telatinib
332012-40-5
C
2
0
H
1
6
ClN
5
O
3
Ceritinib
1032900-25-6
C
2
8
H
3
6
ClN
5
O
3
S
Olmutinib
1353550-13-6
C
2
6
H
2
6
N
6
O
2
S
Radotinib
926037-48-1
C
2
7
H
2
1
F
3
N
8
O
Anlotinib
1058156-90-3
C
2
3
H
2
2
FN
3
O
3
Pyrotinib
1269662-73-8
Nilotinib
Olmutinib
1802181-20-9
Allitinib
897383-62-9
C
2
4
H
1
8
ClFN
4
O
2
Tucatinib
937263-43-9
C
2
6
H
2
4
N
8
O
2
Epertinib
908305-13-5
Famitinib
1044040-56-3
Bozitinib
1440964-89-5
Capmatinib
1029712-80-8
C
2
3
H
1
7
FN
6
O
Mubritinib
366017-09-6
C
2
5
H
2
3
F
3
N
4
O
2
Filgotinib
1206161-97-8
C
2
1
H
2
3
N
5
O
3
S
R-Afatinib
439081-17-1
C
2
4
H
2
5
ClFN
5
O
3
Trametinib
871700-17-3
C
2
6
H
2
3
FIN
5
O
4
Tandutinib
387867-13-2
C
3
1
H
4
2
N
6
O
4
Tivantinib
905854-02-6
C
2
3
H
1
9
N
3
O
2
Golvatinib
928037-13-2
C
3
3
H
3
7
F
2
N
7
O
4
Crizotinib
877399-52-5
C
2
1
H
2
2
Cl
2
FN
5
O
Canertinib
267243-28-7
C
2
4
H
2
5
ClFN
5
O
3
Rebastinib
1020172-07-9
C
3
0
H
2
8
FN
7
O
3
Pexmetinib
1073667-64-7
Flumatinib
895519-90-1
C
2
9
H
2
9
F
3
N
8
O
Pacritinib
937272-79-2
C
2
8
H
3
2
N
4
O
3
Poziotinib
1092364-38-9
C
2
3
H
2
1
Cl
2
FN
4
O
3
Linsitinib
867160-71-2
C
2
6
H
2
3
N
5
O
Varlitinib
845272-21-1
C
2
2
H
1
9
ClN
6
O
2
S
Lenvatinib
417716-92-8
C
2
1
H
1
9
ClN
4
O
4
Amuvatinib
850879-09-3
C
2
3
H
2
1
N
5
O
3
S
Fedratinib
936091-26-8
C
2
7
H
3
6
N
6
O
3
S
Defactinib
1073154-85-4
C
2
0
H
2
1
F
3
N
8
O
3
S
Sulfatinib
1816307-67-1
Glesatinib
936694-12-1
C
3
1
H
2
7
F
2
N
5
O
3
S
2
Canertinib
289499-45-2
C
2
4
H
2
7
Cl
3
FN
5
O
3
Ensartinib
1370651-20-9
C
2
6
H
2
7
Cl
2
FN
6
O
3
Itacitinib
1334298-90-6
C
2
6
H
2
3
F
4
N
9
O
Brigatinib
1197953-54-0
Pexmetinib
945614-12-0
C
3
1
H
3
3
FN
6
O
3
Nazartinib
1508250-71-2
C
2
6
H
3
1
ClN
6
O
2
Naquotinib
1448232-80-1
Solcitinib
1206163-45-2
Sulfatinib
1308672-74-3
Defactinib
1345713-71-4
Lazertinib
1903008-80-9
Poseltinib
1353552-97-2
Edicotinib
1142363-52-7
Ningetinib
1394820-69-9
Glumetinib
1642581-63-2
R-Afatinib
945553-91-3
Lorlatinib
1454846-35-5
C
2
1
H
1
9
FN
6
O
2
Trametinib
1187431-43-1
C
2
6
H
2
3
FIN
5
O
4
.C
2
H
6
OS
Roblitinib
1708971-55-4
Gandotinib
1229236-86-5
C
2
3
H
2
5
ClFN
7
O
Ripretinib
1442472-39-0
Filgotinib
848416-07-9
Glesatinib
1123838-51-6
Sorafetinib
Saracatinib
379231-04-6
C
2
7
H
3
2
ClN
5
O
5
Ulixertinib
869886-67-9
C
2
1
H
2
2
Cl
2
N
4
O
2
Refametinib
923032-37-5
C
1
9
H
2
0
F
3
IN
2
O
5
S
Mereletinib
1421373-65-0
C
2
8
H
3
3
N
7
O
2
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